| Others | 30000 nM | Brain adenylate cyclase 1 | Q08828 | |
| Kd | 45000 nM | Adenosine A1 receptor | P30542 | |
| Ki | 49000 nM | Adenosine A1 receptor | P30542 | |
| Ki | 18100 nM | Adenosine A2a receptor | P29274 | |
| Others | 9 % | Adenosine A3 receptor | P0DMS8 | |
| Ki | 49000 nM | Adenosine A1 receptor | P30542 | |
| Ki | 18100 nM | Adenosine A2a receptor | P29274 | |
| Ki | 100000 nM | Adenosine A3 receptor | P0DMS8 | |
| Others | -1.4 % | Solute carrier family 22 member 1 | O15245 | |
| Ki | 3600000 nM | Monoamine oxidase B | P27338 | |
| Ki | 33800 nM | Adenosine A2b receptor | P29275 | |
| Ki | 10400 nM | Adenosine A2b receptor | P29275 | |
| Others | 9 % | Adenosine A3 receptor | P0DMS8 | |
| Ki | 18100 nM | Adenosine A2a receptor | P29274 | |
| Ki | 49000 nM | Adenosine A1 receptor | P30542 | |
| Ki | 100000 nM | Adenosine A3 receptor | P0DMS8 | |
| Ki | 33800 nM | Adenosine A2b receptor | P29275 | |
| Ki | 10400 nM | Adenosine A2b receptor | P29275 | |
| Potency | 79432.8 nM | DNA polymerase beta | P06746 | |
| IC50 | 4897.79 nM | HERG | Q12809 | |
| Potency | 10000 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
| Potency | 5011.9 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
| Potency | 1412.5 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
| Potency | 44668.4 nM | Chromobox protein homolog 1 | P83916 | |
| Ki | 5011.87 nM | Adenosine A2a receptor | P29274 | |
| Kd | 25118.86 nM | Adenosine A2a receptor | P29274 | |
| Potency | 231.1 nM | Geminin | O75496 | |
| Ki | 44900 nM | Adenosine A1 receptor | P30542 | |
| Ki | 23400 nM | Adenosine A2a receptor | P29274 | |
| Ki | 20500 nM | Adenosine A2b receptor | P29275 | |
| Ki | 100000 nM | Adenosine A3 receptor | P0DMS8 | |
| Others | 3.2 % | Solute carrier organic anion transporter family member 2B1 | O94956 | |
| Others | 22.1 % | Solute carrier organic anion transporter family member 1B3 | Q9NPD5 | |
| Others | -1.8 % | Solute carrier organic anion transporter family member 1B1 | Q9Y6L6 | |
| Others | 72.7 % | Serum albumin | P02768 | |
| Others | 58.4 % | Serum albumin | P02768 | |
| Ki | 44000 nM | Adenosine A1 receptor | P30542 | |
| Ki | 23400 nM | Adenosine A2a receptor | P29274 | |
| IC50 | 50000 nM | Butyrylcholinesterase | P06276 | |
| IC50 | 7250 nM | Acetylcholinesterase | P22303 | |
| Ki | 9560 nM | Adenosine A2a receptor | P29274 | |
| Ki | 2480 nM | Adenosine A2a receptor | P29274 | |
| Ki | 13300 nM | Adenosine A3 receptor | P0DMS8 | |
| Ki | 33800 nM | Adenosine A2b receptor | P29275 | |
| Ki | 23400 nM | Adenosine A2a receptor | P29274 | |
| Ki | 44900 nM | Adenosine A1 receptor | P30542 | |
| Ki | 13300 nM | Adenosine A3 receptor | P0DMS8 | |
| Ki | 23400 nM | Adenosine A2a receptor | P29274 | |
| Ki | 44900 nM | Adenosine A1 receptor | P30542 | |
| Ki | 33800 nM | Adenosine A2b receptor | P29275 | |
| IC50 | 75000 nM | PI3-kinase p110-delta subunit | O00329 | |
| IC50 | 400000 nM | PI3-kinase p110-alpha subunit | P42336 | |
| IC50 | 400000 nM | PI3-kinase p110-beta subunit | P42338 | |
| IC50 | 1000000 nM | PI3-kinase p110-gamma subunit | P48736 | |
| Ki | 20500 nM | Adenosine A2b receptor | P29275 | |
| Ki | 23400 nM | Adenosine A2a receptor | P29274 | |
| Ki | 44900 nM | Adenosine A1 receptor | P30542 | |
| IC50 | 3630000 nM | PI3-kinase p110-gamma subunit | P48736 | |
| Others | 10 % | Cytochrome P450 1A2 | P05177 | |
| Others | 10 % | Cytochrome P450 2B6 | P20813 | |
| Others | 10 % | Cytochrome P450 2C8 | P10632 | |
| Others | 10 % | Cytochrome P450 2C9 | P11712 | |
| Others | 10 % | Cytochrome P450 2C19 | P33261 | |
| Others | 10 % | Cytochrome P450 2D6 | P10635 | |
| Others | 10 % | Cytochrome P450 3A4 | P08684 | |
| Ki | 3800000 nM | Monoamine oxidase B | P27338 | |
| Ki | 33800 nM | Adenosine A2b receptor | P29275 | |
