IC50 | 17000 nM | Phosphodiesterase 2A | O00408 | |
Others | 88.2 % | Acetylcholinesterase | P22303 | |
Others | 46.4 % | Acetylcholinesterase | P22303 | |
IC50 | 24330 nM | Acetylcholinesterase | P22303 | |
Ki | 279 nM | Phosphodiesterase 3A | Q14432 | |
Ki | 417 nM | Phosphodiesterase 3B | Q13370 | |
Others | 118.2 % | Sphingomyelin phosphodiesterase | P17405 | |
Others | 66.3 % | Solute carrier family 22 member 1 | O15245 | |
IC50 | 56.9 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 76 nM | Phosphodiesterase 10A | Q9Y233 | |
Potency | 1995.3 nM | Prelamin-A/C | P02545 | |
Potency | 10000 nM | Nuclear factor NF-kappa-B p105 subunit | P19838 | |
Potency | 91999.7 nM | Ras-related protein Rab-9A | P51151 | |
Potency | 7943.3 nM | Survival motor neuron protein | Q16637 | |
Potency | 12589.3 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 5011.9 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 3162.3 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 10000 nM | Cytochrome P450 2C19 | P33261 | |
Potency | 3981.1 nM | Cytochrome P450 2C19 | P33261 | |
Potency | 5011.9 nM | Cytochrome P450 2C19 | P33261 | |
Potency | 10000 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 2511.9 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 3548.1 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 15848.9 nM | CREB-binding protein | Q92793 | |
Potency | 10000 nM | CREB-binding protein | Q92793 | |
Potency | 39810.7 nM | Arachidonate 15-lipoxygenase | P16050 | |
Potency | 10000 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 2511.9 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 7079.5 nM | Arachidonate 12-lipoxygenase | P18054 | |
Potency | 31622.8 nM | MAP kinase ERK2 | P28482 | |
Potency | 7943.3 nM | MAP kinase ERK2 | P28482 | |
Potency | 10000 nM | Nuclear factor NF-kappa-B p105 subunit | P19838 | |
Potency | 12589.3 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 12589.3 nM | Ubiquitin carboxyl-terminal hydrolase 2 | O75604 | |
Potency | 7943.3 nM | CREB-binding protein | Q92793 | |
Potency | 7943.3 nM | CREB-binding protein | Q92793 | |
Potency | 5011.9 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 707.9 nM | CREB-binding protein | Q92793 | |
Potency | 562.3 nM | CREB-binding protein | Q92793 | |
Potency | 12589.3 nM | Thrombopoietin | P40225 | |
Potency | 2511.9 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 10000 nM | Cytochrome P450 2D6 | P10635 | |
Potency | 12589.3 nM | Cytochrome P450 2D6 | P10635 | |
Potency | 1995.3 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 25118.9 nM | Cytochrome P450 2D6 | P10635 | |
Potency | 2511.9 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 39810.7 nM | Cytochrome P450 2C9 | P11712 | |
Potency | 1258.9 nM | CREB-binding protein | Q92793 | |
Potency | 1258.9 nM | CREB-binding protein | Q92793 | |
Potency | 12589.3 nM | Cytochrome P450 2C9 | P11712 | |
Potency | 1995.3 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 12589.3 nM | Thrombopoietin | P40225 | |
IC50 | 17 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 7244.36 nM | HERG | Q12809 | |
Potency | 7307.8 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
Potency | 5623.4 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Potency | 707.9 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Potency | 6 nM | Chromobox protein homolog 1 | P83916 | |
IC50 | 21 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 36 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 210 nM | Phosphodiesterase 10A | Q9Y233 | |
Others | 13.3 % | Bile acid receptor FXR | Q96RI1 | |
IC50 | 36 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 36 nM | Phosphodiesterase 10A | Q9Y233 | |
IC50 | 92.3 nM | Phosphodiesterase 10A | Q9Y233 | |