IC50 | 75.7 nM | Estrogen receptor alpha | P03372 | |
IC50 | 75.7 nM | Estrogen receptor alpha | P03372 | |
IC50 | 18.6 nM | Estrogen receptor beta | Q92731 | |
IC50 | 18.6 nM | Estrogen receptor beta | Q92731 | |
Others | 5.5 % | 3-keto-steroid reductase | P56937 | |
Others | 2.3 % | 3-keto-steroid reductase | P56937 | |
Potency | 14125.4 nM | Prelamin-A/C | P02545 | |
Potency | 100000 nM | Thyroid hormone receptor beta-1 | P10828 | |
Potency | 31622.8 nM | ATP-dependent DNA helicase Q1 | P46063 | |
Potency | 22387.2 nM | ATP-dependent DNA helicase Q1 | P46063 | |
Potency | 10000 nM | Lysine-specific demethylase 4D-like | B2RXH2 | |
Potency | 56234.1 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 50118.7 nM | Thyroid hormone receptor beta-1 | P10828 | |
Potency | 14125.4 nM | Microtubule-associated protein tau | P10636 | |
Potency | 10000 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 25118.9 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 35481.3 nM | Lysosomal alpha-glucosidase | P10253 | |
Potency | 10000 nM | Hypoxia-inducible factor 1 alpha | Q16665 | |
Potency | 28183.8 nM | 15-hydroxyprostaglandin dehydrogenase [NAD+] | P15428 | |
Potency | 31622.8 nM | Alpha-galactosidase A | P06280 | |
Potency | 28183.8 nM | Bloom syndrome protein | P54132 | |
Potency | 31622.8 nM | Lysosomal alpha-glucosidase | P10253 | |
Potency | 35481.3 nM | DNA polymerase beta | P06746 | |
Potency | 31622.8 nM | Lysosomal alpha-glucosidase | P10253 | |
Potency | 32642.7 nM | ATPase family AAA domain-containing protein 5 | Q96QE3 | |
Potency | 39810.7 nM | Nuclear factor NF-kappa-B p105 subunit | P19838 | |
Potency | 16360.1 nM | Geminin | O75496 | |
Potency | 50118.7 nM | Aryl hydrocarbon receptor | P35869 | |
Potency | 54482.7 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
IC50 | 32340 nM | Rac GTPase-activating protein 1 | Q9H0H5 | |
IC50 | 66600 nM | Small ubiquitin-related modifier 1 | P63165 | |
Potency | 7943.3 nM | Glutaminase kidney isoform, mitochondrial | O94925 | |
Potency | 79432.8 nM | Werner syndrome ATP-dependent helicase | Q14191 | |
IC50 | 14700 nM | Small ubiquitin-related modifier 1 | P63165 | |
Others | -41.5 % | Solute carrier organic anion transporter family member 2B1 | O94956 | |
Others | -21.1 % | Solute carrier organic anion transporter family member 1B3 | Q9NPD5 | |
Others | 73.2 % | Solute carrier organic anion transporter family member 1B1 | Q9Y6L6 | |
IC50 | 12000 nM | Pregnane X receptor | O75469 | |