IC50 | 27600 nM | Leukocyte adhesion molecule-1 | P14151 | |
IC50 | 19100 nM | P-selectin | P16109 | |
IC50 | 500000 nM | Selectin E | P16581 | |
IC50 | 97.3 ug/ml | Aldose reductase | P15121 | |
Ki | 7030 nM | Carbonic anhydrase XIV | Q9ULX7 | |
Ki | 7780 nM | Carbonic anhydrase XII | O43570 | |
Ki | 6990 nM | Carbonic anhydrase IX | Q16790 | |
Ki | 6070 nM | Carbonic anhydrase VII | P43166 | |
Ki | 6130 nM | Carbonic anhydrase VI | P23280 | |
Ki | 9970 nM | Carbonic anhydrase VB | Q9Y2D0 | |
Ki | 4080 nM | Carbonic anhydrase VA | P35218 | |
Ki | 9800 nM | Carbonic anhydrase IV | P22748 | |
Ki | 7490 nM | Carbonic anhydrase III | P07451 | |
Ki | 2250 nM | Carbonic anhydrase II | P00918 | |
Ki | 3200 nM | Carbonic anhydrase I | P00915 | |
Potency | 281.8 nM | Prelamin-A/C | P02545 | |
Potency | 19952.6 nM | Endoplasmic reticulum-associated amyloid beta-peptide-binding protein | Q99714 | |
Potency | 354.8 nM | Lysine-specific demethylase 4D-like | B2RXH2 | |
Potency | 25118.9 nM | Glyceraldehyde-3-phosphate dehydrogenase liver | P04406 | |
Potency | 15848.9 nM | Survival motor neuron protein | Q16637 | |
Potency | 2511.9 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 1000 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 1258.9 nM | Microtubule-associated protein tau | P10636 | |
Potency | 8912.5 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 1995.3 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 1995.3 nM | Microtubule-associated protein tau | P10636 | |
Potency | 25118.9 nM | MAP kinase ERK2 | P28482 | |
Potency | 22387.2 nM | MAP kinase ERK2 | P28482 | |
Potency | 7079.5 nM | 15-hydroxyprostaglandin dehydrogenase [NAD+] | P15428 | |
Potency | 50.1 nM | Endoplasmic reticulum-associated amyloid beta-peptide-binding protein | Q99714 | |
Potency | 12589.3 nM | Cellular tumor antigen p53 | P04637 | |
Potency | 10000 nM | Cellular tumor antigen p53 | P04637 | |
Potency | 39810.7 nM | Histone acetyltransferase GCN5 | Q92830 | |
Potency | 31622.8 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 1995.3 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Others | 0 pm/min/mg | UDP-glucuronosyltransferase 1-1 | P22309 | |
Others | 63.71 % | Estrogen receptor alpha | P03372 | |
Others | 92.19 % | Estrogen receptor alpha | P03372 | |
Potency | 4216.3 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
Potency | 10000 nM | Glutaminase kidney isoform, mitochondrial | O94925 | |
Potency | 47307.9 nM | Interleukin-8 | P10145 | |
Others | 38.9 % | ADAM17 | P78536 | |
Others | 43.5 % | ADAM17 | P78536 | |
Others | 47.9 % | ADAM17 | P78536 | |
Others | 112.2 % | Cytochrome P450 19A1 | P11511 | |
IC50 | 60 nM | Alpha-(1,3)-fucosyltransferase 7 | Q11130 | |
IC50 | 14000 nM | Fucosyltransferase 4 | P22083 | |
Others | 103.1 % | Isocitrate dehydrogenase [NADP] cytoplasmic | O75874 | |
Others | 97.4 % | Isocitrate dehydrogenase [NADP] cytoplasmic | O75874 | |